Lehrstuhl für Pharmazeutische Chemie

Structure-guided development of dual ß2 adrenergic/dopamine D-2 receptor agonists (2016) Weichert D, Stanek M, Hübner H, Gmeiner P Journal article, Original article Spontaneous butenolide ring formation of pregnane-21-O-malonyl hemiesters under mild reaction conditions is facilitated by the 14β-hydroxy group present in all natural cardenolides (2016) Maia de Pádua R, Meitinger N, Hennemann M, Schebitz P, Waibel R, Löber S, Gmeiner P, et al. Journal article, Original article Development of Covalent Ligand-Receptor Pairs to Study the Binding Properties of Nonpeptidic Neurotensin Receptor 1 Antagonists. (2016) Kling R, Plomer M, Lang C, Banerjee A, Hübner H, Gmeiner P Journal article, Original article Mimicking of Arginine by Functionalized N(ω)-Carbamoylated Arginine As a New Broadly Applicable Approach to Labeled Bioactive Peptides: High Affinity Angiotensin, Neuropeptide Y, Neuropeptide FF, and Neurotensin Receptor Ligands As Examples. (2016) Keller M, Kuhn KK, Einsiedel J, Hübner H, Biselli S, Mollereau C, Wifling D, et al. Journal article, Original article Discovery and Characterization of Biased Allosteric Agonists of the Chemokine Receptor CXCR3. (2016) Lampros M, Brox R, Frank T, Poklukar G, Palmisano R, Waibel R, Einsiedel J, et al. Journal article Comparative MD Simulations Indicate a Dual Role for Arg132(3.50) in Dopamine-Dependent D2R Activation (2016) Kling R, Clark T, Gmeiner P Journal article, Original article Development of Photoactivatable Allosteric Modulators for the Chemokine Receptor CXCR3 (2016) Admas T, Bernat V, Heinrich M, Tschammer N Journal article, Original article Structure-guided development of heterodimer-selective GPCR ligands (2016) Hübner H, Schellhorn T, Gienger M, Schaab C, Kaindl J, Leeb L, Clark T, et al. Journal article, Original article Optimization and synthesis of an 18F-labeled dopamine D3 receptor ligand using [18F]fluorophenylazocarboxylic tert-butylester (2016) Nebel N, Maschauer S, Hocke C, Hübner H, Gmeiner P, Prante O Journal article, Original article Attenuation of chemokine receptor function and surface expression as an immunomodulatory strategy employed by human cytomegalovirus is linked to vGPCR US28 (2016) Frank T, Reichel A, Larsen O, Stilp AC, Rosenkilde MM, Stamminger T, Ozawa T, Tschammer N Journal article