Lehrstuhl für Pharmazeutische Chemie

Novel triazolopeptides: chirospecific synthesis and conformational studies of proline derived analogs (2009) Paul A, Einsiedel J, Waibel R, Heinemann FW, Meyer K, Gmeiner P Journal article, Original article A simple chemical method for synthesizing malonyl hemiesters of 21-hydroxy-pregnanes, potential intermediates in cardenolide biosynthesis. (2008) Maia de Pádua R, Waibel R, Kuate SP, Schebitz P, Hahn S, Gmeiner P, Kreis W Journal article, Original article Peptide backbone modifications on the C-terminal hexapeptide of neurotensin (2008) Einsiedel J, Hübner H, Hervet M, Härterich S, Koschatzky S, Gmeiner P Journal article Novel Insights into GPCR-Peptide Interactions: Mutations in Extracellular Loop 1, Ligand Backbone Methylations and Molecular Modeling of Neurotensin Receptor 1 (2008) Härterich S, Koschatzky S, Einsiedel J, Gmeiner P Journal article Novel D3 Selective Dopaminergics Incorporating Enyne Units as Nonaromatic Catechol Bioisosteres: Synthesis, Bioactivity, and Mutagenesis Studies (2008) Doerfler M, Tschammer N, Hamperl K, Hübner H, Gmeiner P Journal article Proline derived spirobarbiturates as highly effective β-turn mimetics incorporating polar and functionalizable constraint elements (2008) Lomlim L, Einsiedel J, Heinemann FW, Meyer K, Gmeiner P Journal article, Original article Structural Characterisation of the E. coli Heat Stable Enterotoxin STh (2008) Matecko I, Burmann BM, Schweimer K, Kalbacher H, Einsiedel J, Gmeiner P, Rösch P Journal article Characterization of the Molecular Fragment that is Responsible for Agonism of Pergolide at Serotonin 5-HT2B and 5-HT2A Receptors (2008) Goernemann T, Hübner H, Gmeiner P, Horowski R, Latte KP, Flieger M, Pertz HH Journal article 18F-Labeled FAUC 346 and BP 897 Derivatives as Subtype-Selective Potential PET Radioligands for the Dopamine D3 Receptor (2008) Hocke C, Prante O, Salama I, Hübner H, Löber S, Kuwert T, Gmeiner P Journal article Synthesis, Radiofluorination and In Vitro Evaluation of Pyrazolo[1,5-a]pyridine Based Dopamine D4 Receptor Ligands: Discovery of an Inverse Agonist Radioligand for PET (2008) Prante O, Tietze R, Hocke C, Löber S, Hübner H, Kuwert T, Gmeiner P Journal article