Lehrstuhl für Pharmazeutische Chemie

Computational Characterization of the Binding Properties of the HIV1-Neutralizing Antibody PG16 and Design of PG16-Derived CDRH3 Peptides (2023) Deubler M, Weißenborn L, Leukel S, Horn A, Eichler J, Sticht H Journal article Therapeutic antagonism of the neurokinin 1 receptor in endosomes provides sustained pain relief (2023) Hegron A, Peach CJ, Tonello R, Seemann P, Teng S, Latorre R, Hübner H, et al. Journal article Inhibiting a promiscuous GPCR: iterative discovery of bitter taste receptor ligands (2023) Fierro F, Peri L, Hübner H, Tabor-Schkade A, Waterloo L, Löber S, Pfeiffer T, et al. Journal article Discovery of 2-Aminopyrimidines as Potent Agonists for the Bitter Taste Receptor TAS2R14 (2023) Waterloo L, Hübner H, Fierro F, Pfeiffer T, Brox R, Löber S, Weikert D, et al. Journal article Phosphoproteomic Analysis of Dopamine D2 Receptor Signaling Reveals Interplay of G Protein- and β-Arrestin-Mediated Effects (2023) Wenk D, Khan S, Ignatchenko V, Hübner H, Gmeiner P, Weikert D, Pischetsrieder M, Kislinger T Journal article Visible-Light-Mediated Radical Arylations Using a Fluorescein- Derived Diazonium Salt: Reactions Proceeding via an Intramolecular Forth and Back Electron Transfer (2023) Diesendorf N, Wenisch P, Oppl J, Heinrich M Journal article Bind&Bite: covalently stabilized heterodimeric coiled-coil peptides for the site-selective, cysteine-free chemical modification of proteins (2023) Beutel J, Tannig P, Di Vincenzo R, Schumacher T, Überla K, Eichler J Journal article Fluorescent Ligands Enable Target Engagement Studies for the Intracellular Allosteric Binding Site of the Chemokine Receptor CXCR2 (2023) Huber M, Wurnig S, Toy L, Weiler C, Merten N, Kostenis E, Hansen FK, Schiedel M Journal article Exploring Structural Determinants of Bias among D4 Subtype-Selective Dopamine Receptor Agonists (2023) Graßl F, Bock L, Huete-Huerta González Á, Schiller M, Gmeiner P, König J, Fromm M, et al. Journal article Tuning the Polarity of Antibiotic-Cy5 Conjugates Enables Highly Selective Labeling of Binding Sites (2023) Graßl F, Konrad M, Krüll J, Pezerovic A, Zähnle L, Burkovski A, Heinrich M Journal article